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程民井

发布时间:2026-01-21 发布单位:


        程民井男,博士,副研究员、博士生导师。20146月毕业于江西中医药大学WilliamHill,获学士学位。20206月毕业于威廉williamhill中药化学专业,获博士学位。20207月进入威廉williamhill中西医结合博士后流动站进行博士后研究。20237月任职于WilliamHill,从事教学科研工作。

        研究方向为天然生物活性小分子和多肽的合成与结构修饰研究。先后主持主持国家自然科学基金面上项目和青年项目(C类)、广东省自然科学基金面上项目等科研项目5项。已发表SCI论文23篇,其中以第一作者或通讯作者在国际权威期刊JACSAngewNat. Commun.Chem. Sci.Org. Lett.Org. Chem. Front. Biochem. Pharmacol. 等杂志发表论文13篇。申请国内外发明专利12项(获授权8项),PCT专利1项,部分专利成果已成功转化。


主持的科研项目:

       [1] 国家自然科学基金面上项目(项目编号:82473801,主持)

       [2] 国家自然科学基金青年科学基金项目(项目编号:82104019,主持)

       [3] 广东省自然科学基金面上项目(项目编号:2025A1515011064,主持)

       [4] 广州市基础研究计划优秀博士启航项目(项目编号:2025A04J3399,主持)

       [5] 中国博士后科学基金面上项目(项目编号:2021M691260,主持)


代表性论文:

        [1] Cheng Min-Jing#, Zhong Li-Ping#, Gu Chen-Chen, Zhu Xu-Jiang, Chen Bo, Liu Jun-Shan, Wang Lei*, Ye Wen-Cai*, Li Chuang-Chuang*. Asymmetric total synthesis of bufospirostenin A. Journal of the American Chemical Society, 2020, 142(42): 12602-12607. (A1-1区,TOP 期刊,IF = 14.612)

        [2] YangChao#, LeiXueping#,*, ChenXian-Bo#, Li Ni-Ping#, LiBoyin, HeYu-Xin, LinShi-Lin, ChenMing, ZhangTian-Hong, WangYong-Heng, GaoHao, LiChuang-Chuang, ChengMin-Jing*, YeWen-Cai*, WangLei*. JACS2025, 2025, 147(29): 38390. (A1-1区,TOP 期刊,IF = 15.7)

        [3] Cheng Min-Jing#, Wu Yan-Yi#, Zeng Hao#, Zhang Tian-Hong, Hu Yan-Xia, Liu Shi-Yi, Cui Rui-Qin, Hu Chun-Xia, Zou Quan-Ming*, Li Chuang-Chuang*, Ye Wen-Cai*, Huang Wei*, Wang Lei*. Asymmetric total synthesis of polycyclic xanthenes and discovery of the first WalK activator with potent activity against MRSA. Nature Communications, 2024, 15: 5879. (A1-1区,TOP 期刊,IF = 14.7)

        [4] Lin Shi-Lin#, Zhao Fen#, Wei Fen#, Shi Ying-Tong, Wen Jing-Kai, Yang Chao, Zhang Hao-Shuo, Li Chuang-Chuang, Liu Chang*, Ye Wen-Cai*,Cheng Min-Jing*, Wang Lei*. Visible-light photocatalyzed skeletal rearrangement enables the synthesis of highly functionalized xanthenes with antitumor activity. Angewandte Chemie International Edition, 2025, e202420671. (A1-1区,TOP 期刊,IF = 16.9)

        [5] Cheng Min-Jing, Cao Jia-Qing, Yang Xin-Yi, Zhong Li-Ping, Hu Li-Jun, Lu Xi, Hou Bao-Long, Hu Ya-Jian, Wang Ying, You Xue-Fu, Wang Lei, Ye Wen-Cai, Li Chuang-Chuang. Catalytic asymmetric total syntheses of myrtucommuacetalone, myrtucommuacetalone B, and callistrilones A, C, D and E. Chemical Science, 2018, 9(6):1488-1495. (A1-1区,TOP 期刊,IF = 9.556)

        [6] HuangQian#, LiNi-Ping#,LinKai#, WangJia-Min, WuZhen-Long, WangWen-Jing, CaoJia-Qing, WangZhen, TuZheng-Chao, Cheng Min-Jing*, YeWen-Cai*, WangLei*. Discovery and Biomimetic syntheses of phloroglucinol-monoterpene-triketone hybrids from Chamelaucium uncinatum with hypoglycemic activity. Organic Letters, 2025, 27(24):6264-6270. (A1-1区,TOP 期刊,IF = 5.0)

        [7] Cheng Min-Jing#, Yang Xin-Yi#, Cao Jia-Qing, Chao Liu, Zhong Li-Ping, Hu Ya-Jian, Wang Ying, You Xue-Fei, Li Chuang-Chuang*, Wang Lei*, Ye Wen-Cai*. Isolation, structure elucidation, and total synthesis of myrtuspirone A from Myrtus communis. Organic Letters, 2019, 21(6):1583-1587. (A1-1区,TOP 期刊,IF = 6.091)

        [8] Zeng Huan#, Cheng Min-Jing#, Liu Jing-Yi, Hu Chun-Xia, Lin Shi-Lin, Cui Rui-Qin, Li Hai-Bo*, Ye Wen-Cai*, Wang Lei*, Huang Wei*. Pyrimirhodomyrtone inhibits Staphylococcus aureus by affecting the activity of NagA. Biochemical Pharmacology, 2023, 210: 115455. (A1-2区,TOP 期刊,IF = 5.8)

        [9] Hu Li-Jun#,Cheng Min-Jing#, Cao Jia-Qing, Zhong Li-Ping, Hu Ya-Jian, Wang Ying, Wang Lei, Ye Wen-Cai, Li Chuang-Chuang. Asymmetric total syntheses of callistrilones B, G and J. Organic Chemistry Frontiers, 2018, 5(9):1506-1510.(A1-1区,TOP 期刊,IF = 5.445)

        [10] Long Xiong-En, Xing Hailiang, He Yixin, Meng Xuanli, Ma Yanling, Liu Chang, Cao Xi, Nan Huiru, Cheng Min-Jing*, Yan Jia-Lei, Liu Junyang. Total synthesis and biological evaluation of Koshidacin B, TAN-1746, and Ac-TAN-1746. BMC Chemistry, 2025, 19: 213.(A1-2区,IF = 4.6)

        [11] GuoHong#, QiMing-Fang#, WangSi-Si, ZhuYa-Hang, LinShi-Lin, ZhengMei-Qi, WuYan-Yi, HuYan-Xia, LiChuang-Chuang, WangLei*,Cheng Min-Jing*, YeWen-Cai*. Biomimetic synthesis of myrtucommulones D-E.The Journal of Organic Chemistry,2025, 90(25): 8737-8744. (A1-2区,IF = 3.2)

        [12] LvNa#, GuChen-Chen#, Xin Zou#, MinLong,*Cheng Min-Jing*, Chuang-Chuang Li. Recent advances in the total synthesis of polycyclic phloroglucinol natural products. Organic Chemistry Frontiers,2026, DOI:10.1039/D5QO01477H.(A1-2区,IF = 4.6)


代表性专利:

       [1] 程民井, 李闯创. 抗菌药物的制备方法, 中国, 2020-1-7, ZL201710338972.5.

       [2] 程民井, 李闯创. 抗菌药物的制备方法, 中国, 2020-12-22, ZL201710338930.1.

       [3] 程民井, 李闯创.抗菌药物的制备方法, 中国, 2021-6-29, ZL201710338022.2.

       [4] 程民井, 钟李平, 顾辰辰, 李闯创. 钠钾ATP酶抑制剂的制备方法, 中国, 2022-09-30, ZL202010242736.5.

       [5] 程民井,叶文才,王磊,杨超,林诗琳,陈明,郑美琪,黄可儿,简健齐,罗钉,张岩,李超. 一种抗菌间苯三酚类化合物及其制备方法与应用, 中国, 2025-11-25, CN202511737025.4.

       [6] 程民井, 叶文才, 王磊, 林凯, 林诗琳, 郭洪, 陈美泓, 曹佳青.多环聚酮类化合物和其制备方法、药物组合物及应用, 中国, 2026-1-6, ZL202411413000.4.

       [7] 王磊, 叶文才, 程民井. 一种间苯三酚衍生物及其在制备抗菌药物中的应用, 2019-07-19, 中国, ZL 201610347417.4.


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联系邮箱:chengmj1235@jnu.edu.cn